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MASTL-IN-1

Chemical Structure : MASTL-IN-1

CAS No.: 1349670-22-9

MASTL-IN-1 (MASTL inhibitor)

Catalog No.: PC-23352Not For Human Use, Lab Use Only.

MASTL-IN-1 is a potent, selective inhibitor of microtubule-associated serine/threonine kinase-like (MASTL, Greatwall) with Ki of 4.4 nM, cellular pENSA IC50 of 23 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

MASTL-IN-1 is a potent, selective inhibitor of microtubule-associated serine/threonine kinase-like (MASTL, Greatwall) with Ki of 4.4 nM, cellular pENSA IC50 of 23 nM.

Physicochemical Properties

M.Wt 430.51
Formula C24H26N6O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

9-methoxy-8-((1-methylpiperidin-4-yl)methoxy)-2-(pyrazin-2-yl)benzo[c][2,7]naphthyridin-4-amine

References

1. Gallego RA, et al. J Med Chem. 2024 Nov 5. doi: 10.1021/acs.jmedchem.4c01659.

2. Patent WO2008109613.

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