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Chemical Structure : MK-3901
Catalog No.: PC-63353Not For Human Use, Lab Use Only.
MK-3901 is a potent, selective, orally active P2X3 antagonist with IC50 of 21 nM.
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MK-3901 is a potent, selective, orally active P2X3 antagonist with IC50 of 21 nM.
MK-3901 demonstrates efficacy similar to that of naproxen, after 60 mg/kg (p.o.) administration with EC90 of approximately 3 uM in the rat CFA model of inflammatory pain.
| M.Wt | 481.531 | |
| Formula | C28H24FN5O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Ginnetti AT, et al. Bioorg Med Chem Lett. 2018 May 1;28(8):1392-1396.
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