MK204 | AKR1B10 inhibitor | Probechem Biochemicals

Chemical Structure : MK204

MK204 (MK-204)

Catalog No.: PC-62883Not For Human Use, Lab Use Only.

MK204 is a potent, selective AKR1B10 inhibitor with IC50 of 80 nM, shows high selective (270-fold) over AKR1B1.

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Biological Activity

MK204 is a potent, selective AKR1B10 inhibitor with IC50 of 80 nM, shows high selective (270-fold) over AKR1B1.
MK204 is a lead compound targeting the distinct AKR1B10 specificity pocket and with a strong X-bond.

Physicochemical Properties

M.Wt	714.221
Formula	C16H9Br5ClNO4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Acetic acid, 2-[5-chloro-2-[[[(2,3,4,5,6-pentabromophenyl)methyl]amino]carbonyl]phenoxy]-

References

1. Cousido-Siah A, et al. ACS Chem Biol. 2016 Oct 21;11(10):2693-2705.

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MK204 (MK-204)

Biological Activity

Physicochemical Properties

References

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