ML753286 ((S)-ML753286)

Chemical Structure : ML753286

CAS No.: 1699720-85-8

Catalog No.: PC-20192Not For Human Use, Lab Use Only.

ML753286 ((S)-ML753286) is a potent, selective BCRP inhibitor with IC50 of 0.6 uM (BCRP efflux transporter), shows no activity against P-glycoprotein (P-gp), organic anion-transporting polypeptide (OATP), or major cytochrome P450s (CYPs).

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5 mg	$428	In stock
10 mg	$728	In stock
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Biological Activity

ML753286 ((S)-ML753286) is a potent, selective BCRP inhibitor with IC50 of 0.6 uM (BCRP efflux transporter), shows no activity against P-glycoprotein (P-gp), organic anion-transporting polypeptide (OATP), or major cytochrome P450s (CYPs).

Physicochemical Properties

M.Wt	355.44
Formula	C20H25N3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(3S,6S,12aS)-6-isobutyl-9-methoxy-3-methyl-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione

References

1. Yuexian Li, et al. Bioorg Med Chem Lett. 2016 Jan 15;26(2):551-555.

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