BCRP (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-20192	ML753286 BCRP inhibitor	ML753286 ((S)-ML753286) is a potent, selective BCRP inhibitor with IC50 of 0.6 uM (BCRP efflux transporter), shows no activity against P-glycoprotein (P-gp), organic anion-transporting polypeptide (OATP), or major cytochrome P450s (CYPs).
PC-43183	YHO-13351 free base ABCG2 inhibitor	YHO-13351 is an orally available prodrug of YHO-13177, which can specifically reverse BCRP/ABCG2-mediated drug resistance in vitro and in vivo.
PC-43182	YHO-13351 ABCG2 inhibitor	YHO-13351 is an orally available prodrug of YHO-13177, which can specifically reverse BCRP/ABCG2-mediated drug resistance in vitro and in vivo.
PC-43181	YHO-13177 ABCG2 inhibitor	YHO-13177 is a acrylonitrile derivative and active form of YHO-13351 that can specifically reverse BCRP/ABCG2-mediated drug resistance in vitro and in vivo.
PC-45706	KS176 BCRP inhibitor	KS176 is a potent and selective inhibitor of BCRP multidrug transporter with IC50 of 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays, respectively.
PC-42054	Ko143 ABCG2 inhibitor	Ko143 is a nontoxic analog of fungal toxin fumitremorgin C and potent, orally bioavailable inhibitor of BCRP (ABCG2) with EC90 of 26 nM.
PC-42127	Brevianamide F BCRP inhibitor	Brevianamide F (Cyclo(L-Pro-L-Trp)) is a naturally occurring 2,5-diketopiperazine that possess interesting breast cancer resistance protein (BCRP) inhibitory activity.

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