MLS1082 | D1 dopamine PAM | Probechem Biochemicals

Chemical Structure : MLS1082

CAS No.: 883958-36-9

MLS1082 (MLS-1082, MLS 1082)

Catalog No.: PC-35534Not For Human Use, Lab Use Only.

MLS1082 is a novel positive allosteric modulator of the D1 dopamine receptor, potentiatse dopamine-stimulated G-protein- and β-arrestin-mediated signaling (EC50=123 nM).

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Biological Activity

MLS1082 is a novel positive allosteric modulator of the D1 dopamine receptor, potentiatse dopamine-stimulated G-protein- and β-arrestin-mediated signaling (EC50=123 nM).
MLS1082 increase the affinity of dopamine for the D1 receptor with low micromolar potencies.

Physicochemical Properties

M.Wt	385.467
Formula	C24H23N3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-cyclohexyl-10-methyl-3-phenylpyrimido[4,5-b]quinoline-4,5(3H,10H)-dione

References

1. Luderman KD, et al. Mol Pharmacol. 2018 Aug 1. pii: mol.118.113175.

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MLS1082 (MLS-1082, MLS 1082)

Biological Activity

Physicochemical Properties

References

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