MMSET-IN-1 |CAS:1998139-29-9 Probechem Biochemicals

Chemical Structure : MMSET-IN-1

MMSET-IN-1 (NSD2 inhibitor 1)

Catalog No.: PC-62409Not For Human Use, Lab Use Only.

MMSET-IN-1 (NSD2 inhibitor 1) is a potent, selective epigenetic oncogene MMSET (aka NSD2 or WHSC1) inhibitor with Ki/IC50 of 1.6/3.3 uM.

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Biological Activity

MMSET-IN-1 (NSD2 inhibitor 1) is a potent, selective epigenetic oncogene MMSET (aka NSD2 or WHSC1) inhibitor with Ki/IC50 of 1.6/3.3 uM.
MMSET-IN-1 shows sub-micromolar inhibition of SETD2 and promising selectivity against a panel of 13 other KMTs.

Physicochemical Properties

M.Wt	423.474
Formula	C18H29N7O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S)-2-amino-6-((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)-5-(propylamino)hexanoic acid

References

1. Tisi D, et al. ACS Chem Biol. 2016 Nov 18;11(11):3093-3105.

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MMSET-IN-1 (NSD2 inhibitor 1)

Biological Activity

Physicochemical Properties

References

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