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Chemical Structure : MRS2500
Catalog No.: PC-61412Not For Human Use, Lab Use Only.
MRS2500 is a highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM.
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MRS2500 is a highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM.
MRS2500 inhibits ADP-induced aggregation of human platelets with IC50 of 0.95 nM.
MRS2500 shows strong antithrombotic activity in mice.
| M.Wt | 561.166 | |
| Formula | C13H18IN5O8P2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Kim HS, et al. J Med Chem. 2003 Nov 6;46(23):4974-87.
2. Hechler B, et al. J Pharmacol Exp Ther. 2006 Feb;316(2):556-63.
3. Gao ZG, et al. Mol Pharmacol. 2017 Sep 1. pii: mol.117.109660.
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