MRS4458 | P2Y14 antagonist | Probechem Biochemicals

Chemical Structure : MRS4458

MRS4458 (MRS 4458, MRS 4458)

Catalog No.: PC-35048Not For Human Use, Lab Use Only.

MRS4458 is a potent, highly specific antagonist of P2Y14 receptor with IC50 of 169 nM, does not display extensive off-target interactions with biogenic amine receptors.

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Biological Activity

MRS4458 is a potent, highly specific antagonist of P2Y14 receptor with IC50 of 169 nM, does not display extensive off-target interactions with biogenic amine receptors.

Physicochemical Properties

M.Wt	515.511
Formula	C24H20F3N5O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)benzoic acid

References

1. Yu J, et al. J Med Chem. 2018 May 16. doi: 10.1021/acs.jmedchem.8b00168.

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MRS4458 (MRS 4458, MRS 4458)

Biological Activity

Physicochemical Properties

References

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