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MRS4478

Chemical Structure : MRS4478

CAS No.: 2225834-59-1

MRS4478 (MRS 4478, MRS-4478)

Catalog No.: PC-35049Not For Human Use, Lab Use Only.

MRS4478 is a potent, highly specific antagonist of P2Y14 receptor with IC50 of 269 nM, does not display extensive off-target interactions with biogenic amine receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    MRS4478 is a potent, highly specific antagonist of P2Y14 receptor with IC50 of 269 nM, does not display extensive off-target interactions with biogenic amine receptors.

    Physicochemical Properties

    M.Wt 452.393
    Formula C23H15F3N4O3
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    4'-Carbamoyl-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol1-yl)-[1,1'-biphenyl]-3-carboxylic acid

    References

    1. Yu J, et al. J Med Chem. 2018 May 16. doi: 10.1021/acs.jmedchem.8b00168.

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