MRS4738 | P2Y14 inhibitor | Probechem Biochemicals

Chemical Structure : MRS4738

Catalog No.: PC-20960Not For Human Use, Lab Use Only.

MRS4738 is a potent, selective antagonist of Gi protein-coupled P2Y14 receptor (P2Y14R, GPR105) with IC50 of 3.11 nM.

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Biological Activity

MRS4738 is a potent, selective antagonist of Gi protein-coupled P2Y14 receptor (P2Y14R, GPR105) with IC50 of 3.11 nM.

M.Wt	487.52
Formula	C30H24F3NO2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C(O)C1=CC(C2=CC=C([C@@H]3[C@@]4([H])CN[C@@](C4)([H])C3)C=C2)=C5C=CC(C6=CC=C(C(F)(F)F)C=C6)=CC5=C1

1. Zhiwei Wen, et al. J Med Chem. 2022 Feb 24;65(4):3434-3459.