MS023 | type I PRMTs inhibitor | Probechem Biochemicals

Chemical Structure : MS023

CAS No.: 1831110-54-3

MS023 (MS-023, MS 023)

Catalog No.: PC-45658Not For Human Use, Lab Use Only.

MS023 is a potent, selective, and cell-active inhibitor of type I PRMTs with IC50s of 30/119/83/4/5 nM for PRMT1/3/4/6/8 respectively.

Packing	Price	Stock
5 mg	$88	In stock
10 mg	$138	In stock
25 mg	$228	In stock
50 mg	$388	In stock
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

MS023 is a potent, selective, and cell-active inhibitor of type I PRMTs with IC50s of 30/119/83/4/5 nM for PRMT1/3/4/6/8 respectively.
MS023 does not inhibit PRMT5/9/7(>10 uM).
MS023 inhibits H4R3me2a and H3R2me2a levels in MCF7 cells.

Physicochemical Properties

M.Wt	287.3999
Formula	C17H25N3O
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	DMSO: ≥ 30 mg/mL
Chemical Name/SMILES	1,2-Ethanediamine, N1-methyl-N1-[[4-[4-(1-methylethoxy)phenyl]-1H-pyrrol-3-yl]methyl]-

References

1. Eram MS, et al. ACS Chem Biol. 2016 Mar 18;11(3):772-81.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

MS023 (MS-023, MS 023)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.