MS4138 | SETD8 inhibitor | Probechem Biochemicals

Chemical Structure : MS4138

MS4138 (MS-4138)

Catalog No.: PC-26273Not For Human Use, Lab Use Only.

MS4138 is a potent, selective and covalent inhibitor of protein lysine methyltransferase (PKMT) SETD8 with IC50 of 1.4 uM, covalently modifies SETD8 at Cys311.

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Biological Activity

MS4138 is a potent, selective and covalent inhibitor of protein lysine methyltransferase (PKMT) SETD8 with IC50 of 1.4 uM, covalently modifies SETD8 at Cys311.

Physicochemical Properties

M.Wt	414.51
Formula	C21H30N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(3-((7-(2-aminoethoxy)-6-methoxy-2-(pyrrolidin-1-yl)quinazolin-4-yl)amino)propyl)acrylamide

References

1. Shi Chen, et al. Elife. 2019 May 13:8:e45403.

2. Patent WO2015172076A1.

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MS4138 (MS-4138)

Biological Activity

Physicochemical Properties

References

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