Chemical Structure : Mapracorat
CAS No.:
887375-26-0
Mapracorat
(ZK 245186, BOL 303242X, BAY865319)
Catalog No. : PC-61603Not For Human Use, Lab Use Only.
Mapracorat (ZK 245186) is a potent, selective and non-steroid glucocorticoid receptor (GR) agonist with binding Ki of 1.9 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6160301
Biological Activity
Mapracorat (ZK 245186) is a potent, selective and non-steroid glucocorticoid receptor (GR) agonist with binding Ki of 1.9 nM.
Physicochemical Properties
M.Wt
462.489
Formula
C25H26F4N2O2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
(2R)-1,1,1-trifluoro-4-(5-fluoro-2,3-dihydro-1-benzofuran-7-yl)-4-methyl-2-[[(2-methylquinolin-5-yl)amino]methyl]pentan-2-ol
References
1. Schäcke H, et al. Br J Pharmacol.
2. Zhang JZ, et al. Mol Vis.
3. Shafiee A, et al. Invest Ophthalmol Vis Sci.
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