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Metopimazine

Chemical Structure : Metopimazine

CAS No.: 14008-44-7

Metopimazine (EXP999, RP9965)

Catalog No.: PC-24638Not For Human Use, Lab Use Only.

Metopimazine is a selective, peripherally restricted dopamine D2 receptor (D2R) antagonist, has potential for the symptomatic treatment of nausea and vomiting and chemotherapy-induced nausea and vomiting.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Metopimazine is a selective, peripherally restricted dopamine D2 receptor (D2R) antagonist, has potential for the symptomatic treatment of nausea and vomiting and chemotherapy-induced nausea and vomiting.

Physicochemical Properties

M.Wt 445.60
Formula C22H27N3O3S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-Piperidinecarboxamide, 1-[3-[2-(methylsulfonyl)-10H-phenothiazin-10-yl]propyl]-

References

1. Busby RW, et al. Pharmacol Res Perspect. 2022 Feb;10(1):e00903.

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