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Mocaciclib

Chemical Structure : Mocaciclib

CAS No.: 2766124-39-2

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Mocaciclib (Q901)

Catalog No.: PC-24960Not For Human Use, Lab Use Only.

Mocaciclib (Q901) is a highly selective and potent CDK7 inhibitor, forms a covalent bond with C312 of the CDK7 C-terminal domain.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Mocaciclib (Q901) is a highly selective and potent CDK7 inhibitor, forms a covalent bond with C312 of the CDK7 C-terminal domain.
Mocaciclib (Q901) demonstrates selective cytotoxic activities in a broad spectrum of solid tumor lineages.
Mocaciclib (Q901) is compound 64 extracted from Patent WO2019197546 A1.

Physicochemical Properties

M.Wt 609.71
Formula C33H36FN9O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Fluoro-N-[1-[2-[[[2-[[[(3R,4R)-3-hydroxy-4-piperidinyl]methyl]amino]-8-(1-methylethyl)pyrazolo[1,5-a]-1,3,5-triazin-4-yl]amino]methyl]phenyl]-6-isoquinolinyl]-2-propenamide

References

1. Patent WO2019197546 A1.

2. Donghoon Yu, et al. Cancer Res (2022) 82 (12_Supplement): 2574.

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