Mpro inhibitor GD-9

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Chemical Structure : Mpro inhibitor GD-9

Catalog No.: PC-49579Not For Human Use, Lab Use Only.

Mpro inhibitor GD-9 is a potent, covalent SARS-CoV-2 main protease (Mpro) inhibitor with IC50 of 0.18 uM, exhibits antiviral potency against SARS-CoV-2 with EC50 of 2.64 uM.

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Biological Activity

Mpro inhibitor GD-9 is a potent, covalent SARS-CoV-2 main protease (Mpro) inhibitor with IC50 of 0.18 uM, exhibits antiviral potency against SARS-CoV-2 with EC50 of 2.64 uM.
GD-9 shows similar antiviral potency to that of remdesivir (EC50 = 2.27 μM).
GD-9 presented favorable target selectivity for SARS-CoV-2 Mpro versus human cysteine proteases.

Physicochemical Properties

M.Wt	446.77
Formula	C18H18Cl3N3O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-4-(2-chloroacetyl)-1-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)piperazine-2-carboxamide

References

1. Gao S, et al. J Med Chem. 2022 Dec 22;65(24):16902-16917.

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