Myokinasib-II

Chemical Structure : Myokinasib-II

Catalog No.: PC-23164Not For Human Use, Lab Use Only.

Myokinasib-II is a potent and highly selective myosin light-chain kinase (MLCK) chemical probe inhibitor with IC50 of 4.4 uM for MLCK-1.

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Biological Activity

Myokinasib-II is a potent and highly selective myosin light-chain kinase (MLCK) chemical probe inhibitor with IC50 of 4.4 uM for MLCK1.
Myokinasib-II displays better potency, better selectivity profile, and no nonspecific interference in relevant assays as compared to other known MLCK inhibitors.

Physicochemical Properties

M.Wt	437.47
Formula	C24H24FN3O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	ethyl (6R,7R,8R,9R)-8-(4-fluoro-2-methylphenyl)-6-methyl-7-nitro-6,7,8,10-tetrahydro-6,9-epiminocyclohepta[b]indole-9(5H)-carboxylate

References

1. Gautam Kumar, et al. ACS Chem Biol. 2024 Sep 20. doi: 10.1021/acschembio.4c00336.

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Myokinasib-II

Biological Activity

Physicochemical Properties

References

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