NAH-C3-GPKK

Chemical Structure : NAH-C3-GPKK

Catalog No.: PC-72717Not For Human Use, Lab Use Only.

NAH-C3-GPKK is a potent, selective protein N-terminal methyltransferase 1 (NTMT1) bisubstrate inhibitor with Kiapp of 7 nM in endogenous proteomes.

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Biological Activity

NAH-C3-GPKK is a potent, selective protein N-terminal methyltransferase 1 (NTMT1) bisubstrate inhibitor with Kiapp of 7 nM in endogenous proteomes.
NAH-C3-GPKK also potently inhibit a methyltransferase complex HemK2-Trm112 (also known as KMT9-Trm112, IC50=0.3 uM).
NAH-C3-GPKK is the first potent inhibitor for HemK2/KMT9.

Physicochemical Properties

M.Wt	835.965
Formula	C36H61N13O10
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES

References

1. Dongxing Chen, et al. ACS Chem Biol. 2021 Jul 16;16(7):1234-1242.

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NAH-C3-GPKK

Biological Activity

Physicochemical Properties

References

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