NSD2 inhibitor PTD2 | NSD2 inhibitor | Probechem Biochemicals

Chemical Structure : NSD2 inhibitor PTD2

NSD2 inhibitor PTD2 (Ac-Gly-Val-Nle-Arg-Ile-NH2)

Catalog No.: PC-28088Not For Human Use, Lab Use Only.

NSD2 inhibitor PTD2 is a peptide derived from histone H4 sequence and inhibitor for the histone methyltransferase WHSC1 (Nuclear receptor-binding SET domain protein 2, NSD2, MMSET) with SPR KD of 3.0 uM, IC50 of 22 uM and 3.2 uM for NSD2 and NSD3 respectively.

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Biological Activity

NSD2 inhibitor PTD2 is a peptide derived from histone H4 sequence and inhibitor for the histone methyltransferase WHSC1 (Nuclear receptor-binding SET domain protein 2, NSD2, MMSET) with SPR KD of 3.0 uM, IC50 of 22 uM and 3.2 uM for NSD2 and NSD3 respectively.
PTD2 demonstrates no enzymatic inhibition against the entire panel of methyltransferases.

Physicochemical Properties

M.Wt	597.76
Formula	C27H51N9O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Sequence: Ac-Gly-Val-Nle-Arg-Ile-NH2

References

1. Morrison MJ, et al. PLoS One. 2018 May 9;13(5):e0197082.

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NSD2 inhibitor PTD2 (Ac-Gly-Val-Nle-Arg-Ile-NH2)

Biological Activity

Physicochemical Properties

References

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