Nardilysin inhibitor R5-1

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Chemical Structure : Nardilysin inhibitor R5-1

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Catalog No.: PC-28094Not For Human Use, Lab Use Only.

Nardilysin inhibitor R5-1 is a small-molecule inhibitor of nardilysin (NRDC), inhibits NRDC activity in a non-competitive manner, attenuates NRDC-dependent transcriptional repression of PGC-1α, phenocopying the effect of catalytic inactivation, significantly ameliorates arthritis severity in mouse model of autoimmune arthritis.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Nardilysin inhibitor R5-1 is a small-molecule inhibitor of nardilysin (NRDC), inhibits NRDC activity in a non-competitive manner, attenuates NRDC-dependent transcriptional repression of PGC-1α, phenocopying the effect of catalytic inactivation, significantly ameliorates arthritis severity in mouse model of autoimmune arthritis.

Physicochemical Properties

M.Wt	234.27
Formula	C11H10N2O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(quinoxalin-2-ylthio)propanoic acid

References

1. Amano Y, et al. Biochem Pharmacol. 2026 Sep 9:118456.

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