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Chemical Structure : OR-S0
Catalog No.: PC-72290Not For Human Use, Lab Use Only.
OR-S0 is a potent, selective EZH2 inhibitor with IC50 of 11 nM, weakly inhibitor EZH1 (IC50=91 nM).
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OR-S0 is a potent, selective EZH2 inhibitor with IC50 of 11 nM, weakly inhibitor EZH1 (IC50=91 nM).
OR-S0 inhibits H3K27me3 in HCT116 cells with IC50 of 24 nM, inhibited the growth of KARPAS‐422 cells in a dose‐dependent manner with GI50 of 210 nM.
| M.Wt | 616.763 | |
| Formula | C34H44N6O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Daisuke Honma, et al. Cancer Sci. 2017 Oct;108(10):2069-2078.
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