Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
    English |     Chinese

Product Inquiry: sales@probechem.com
Order/PO receiving: order@probechem.com

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Cannabinoid Receptor-Olorinab
Olorinab

Chemical Structure : Olorinab

CAS No.: 1268881-20-4

Add to Favorites

Olorinab (APD371, APD-371)

Catalog No.: PC-60146Not For Human Use, Lab Use Only.

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.

Packing Price Stock Quantity
5 mg $128 In stock
10 mg $198 In stock
25 mg $358 In stock
50 mg Get quote
100 mg Get quote
Get Quotation Now
* Please select Quantity before adding items.
 or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.
Olorinab (APD371) displays no activity against CB1 receptors (EC50>10 uM).
Olorinab (APD371) exhibits activity in rat model of osteoarthritis pain.

Physicochemical Properties

M.Wt 357.414
Formula C18H23N5O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

3-((4aS,5aS)-3-(((S)-1-hydroxy-3,3-dimethylbutan-2-yl)carbamoyl)-4,4a,5,5a-tetrahydro-1H-cyclopropa[4,5]cyclopenta[1,2-c]pyrazol-1-yl)pyrazine 1-oxide

References

1. Sangdon Han, et al. ACS Med. Chem. Lett., 2017, 8 (12), pp 1309-1313.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: