Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : Omarigliptin
CAS No.: 1226781-44-7
Catalog No.: PC-44866Not For Human Use, Lab Use Only.
Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $198 | In stock | |
| 50 mg | $298 | In stock | |
| 100 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM.
Omarigliptin (MK-3102) shows high selectivity against QPP, DPP8,FAP (IC50>20 uM).
Omarigliptin (MK-3102) is efficacious in the diabetes PD model and excellent pharmacokinetic profile.
| M.Wt | 398.4275 | |
| Formula | C17H20F2N4O3S | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
2H-Pyran-3-amine, 2-(2,5-difluorophenyl)-5-[2,6-dihydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-, (2R,3S,5R)- |
|
1. Biftu T, et al. Bioorg Med Chem Lett. 2013 Oct 1;23(19):5361-6.
2. Biftu T, et al. J Med Chem. 2014 Apr 24;57(8):3205-12.
3. Burness CB. Drugs. 2015 Nov;75(16):1947-52.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
