Catalog No.: PC-42724Not For Human Use, Lab Use Only.
Otenabant hydrochloride (CP-945598) is a potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively.
Otenabant hydrochloride (CP-945598) is a potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively.
Otenabant hydrochloride has low affinity (Ki=7600 nM) for human CB2 receptors.
Otenabant hydrochloride reverses cannabinoid agonist mediated responses, reduces food intake, and increases energy expenditure and fat oxidation in rodents.
