PBRM1-BD2 inhibitor 34 | PBRM1-BD2 inhibitor

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Chemical Structure : PBRM1-BD2 inhibitor 34

CAS No.: 2819989-75-6

PBRM1-BD2 inhibitor 34 (PBRM1-BD2-IN-8)

Catalog No.: PC-25803Not For Human Use, Lab Use Only.

PBRM1-BD2 inhibitor 34 (PBRM1-BD2-IN-8) is a potent, selective PBRM1 bromodomain inhibitor with Kd of4.4 uM, IC50 of 0.16 uM for PBRM1-BD2, shows promising inhibition toward PBRM1-dependent prostate cancer cell line LNCaP with IC50 of 9 uM.

Packing	Price	Stock
5 mg	$128	In stock
10 mg	$198	In stock
25 mg	$358	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Physicochemical Properties

M.Wt	317.19
Formula	C15H13BrN2O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-Bromo-2-(m-tolyl)-2,3-dihydroquinazolin-4(1H)-one

References

1. Shishodia S, et al. J Med Chem. 2022 Oct 27;65(20):13714-13735.

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PBRM1-BD2 inhibitor 34 (PBRM1-BD2-IN-8)

Biological Activity

Physicochemical Properties

References

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