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Chemical Structure : PD128907 hydrochloride
CAS No.: 300576-59-4
Catalog No.: PC-70058Not For Human Use, Lab Use Only.
PD128907 hydrochloride is a potent, selective and orally active agonist of dopamine D3 receptor (D3R) with Ki of 20 nM.
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|---|---|---|---|
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| 10 mg | $288 | In stock | |
| 25 mg | $458 | In stock | |
| 50 mg | $728 | In stock | |
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PD128907 hydrochloride is a potent, selective and orally active agonist of dopamine D3 receptor (D3R) with Ki of 20 nM.
PD128907 hydrochloride displays 18-200-fold selectivity over other dopamine receptor subtypes.
PD128907 hydrochloride decreases dopamine release both in rat striatum, nucleus accumbens and medial frontal cortex, decreases spontaneous locomotor activity (LMA) in rats; orally active.
| M.Wt | 285.77 | |
| Formula | C14H19NO3.HCl | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
(4aR,10bR)-4-propyl-3,4,4a,10b-tetrahydro-2H,5H-chromeno[4,3-b][1,4]oxazin-9-ol hydrochloride |
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1. DeWald HA, et al. J Med Chem. 1990 Jan;33(1):445-50.
2. Pugsley TA, et al. J Pharmacol Exp Ther. 1995 Dec;275(3):1355-66.
3. Bristow LJ, et al. Neuropharmacology. 1996 Mar;35(3):285-94.
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