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PF-06256142

Chemical Structure : PF-06256142

CAS No.: 1609583-14-3

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PF-06256142 (PF06256142)

Catalog No.: PC-35799Not For Human Use, Lab Use Only.

PF-06256142 (PF06256142) is a potent and selective orthosteric agonist of the D1 receptor with EC50 (cAMP) of 33 nM, shows exquisitely selectivity over D2.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    PF-06256142 (PF06256142) is a potent and selective orthosteric agonist of the D1 receptor with EC50 (cAMP) of 33 nM, shows exquisitely selectivity over D2.
    PF-06256142 demonsrates reduced receptor desensitization relative to dopamine and other catechol-containing agonists.

    Physicochemical Properties

    M.Wt 356.385
    Formula C21H16N4O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (+)-4-(3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy)furo[3,2-c]pyridine

    References

    1. Davoren JE, et al. J Med Chem. 2018 Nov 15. doi: 10.1021/acs.jmedchem.8b01622.

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