Chemical Structure : PF-06462894
Catalog No.: PC-61058Not For Human Use, Lab Use Only.
A potent, subtype-selective mGluR5 negative allosteric modulator with Ki of 6.1 nM.
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
A potent, subtype-selective mGluR5 negative allosteric modulator with Ki of 6.1 nM; possesses favorable properties and a predicted low clinical dose (2 mg twice daily), does not show any evidence of immune activation in a mouse drug allergy model.
M.Wt | 329.4 | |
Formula | C18H23N3O3 | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
1. Stepan AF, et al. J Med Chem. 2017 Sep 28;60(18):7764-7780.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright