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Chemical Structure : PF-219061
Catalog No.: PC-70057Not For Human Use, Lab Use Only.
PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM.
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PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM.
PF-219061 has >1000-fold functional selectivity over D2, displays minimal binding activity (IC50>10 uM) against a wide panel of targets including dopamine D1 and D5 receptors.
PF-219061 demonstrates activity in animal models of male erectile dysfunction.
| M.Wt | 235.327 | |
| Formula | C14H21NO2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Blagg J, et al. Bioorg Med Chem Lett. 2007 Dec 15;17(24):6691-6.
2. Attkins NJ, et al. Xenobiotica. 2009 Jul;39(7):523-33.
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