PF-4840154 | TRPA1 agonist | Probechem Biochemicals

Chemical Structure : PF-4840154

CAS No.: 1332708-14-1

PF-4840154 (PF4840154)

Catalog No.: PC-45556Not For Human Use, Lab Use Only.

PF-4840154 is a potent, selective agonist of the rat (EC50=97 nM) and human (EC50=23 nM) TRPA1 channel.

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Biological Activity

PF-4840154 is a potent, selective agonist of the rat (EC50=97 nM) and human (EC50=23 nM) TRPA1 channel.
PF-4840154 elicitsTRPA1-mediated nocifensive behaviour in mouse.

Physicochemical Properties

M.Wt	466.6189
Formula	C26H38N6O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	5-Pyrimidinecarboxamide, 4-[(2-methylpropyl)amino]-N-(phenylmethyl)-2-[4-[(tetrahydro-2H-pyran-3-yl)methyl]-1-piperazinyl]-

References

1. Ryckmans T, et al. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4857-9.

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PF-4840154 (PF4840154)

Biological Activity

Physicochemical Properties

References

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