PFI-4 | BRPF1 inhibitor | Probechem Biochemicals

Chemical Structure : PFI-4

CAS No.: 900305-37-5

PFI-4 (PFI4, BRPF1 inhibitor PFI-4)

Catalog No.: PC-45507Not For Human Use, Lab Use Only.

PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.

Packing	Price	Stock
10 mg	$58	In stock
25 mg	$98	In stock
50 mg	$148	In stock
100 mg	$238	In stock
250 mg		Get quote

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Biological Activity

PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
PFI-4 exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.

Physicochemical Properties

M.Wt	380.4402
Formula	C21H24N4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: 26 mg/mL
Chemical Name/SMILES	Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxy-

References

1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.

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PFI-4 (PFI4, BRPF1 inhibitor PFI-4)

Biological Activity

Physicochemical Properties

References

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