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PFI-4

Chemical Structure : PFI-4

CAS No.: 900305-37-5

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PFI-4 (PFI4, BRPF1 inhibitor PFI-4)

Catalog No.: PC-45507Not For Human Use, Lab Use Only.

PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.

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10 mg $88 In stock
25 mg $138 In stock
50 mg $218 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
PFI-4 exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.

Physicochemical Properties

M.Wt 380.4402
Formula C21H24N4O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: 26 mg/mL
Chemical Name/SMILES

Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxy-

References

1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.

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