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PK14105

Chemical Structure : PK14105

CAS No.: 107257-28-3

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PK14105 (PK-14105)

Catalog No.: PC-42106Not For Human Use, Lab Use Only.

PK14105 is a potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

PK14105 is a potent photoaffinity ligand for the peripheral-type benzodiazepine binding site with Ki of 4 nM.
PK14105 attaches covalently and specifically to all the PBS when cardiac membranes are irradiated with this compound under ultraviolet light.

Physicochemical Properties

M.Wt 381.4002
Formula C21H20FN3O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
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Solubility

DMSO: ≥ 30 mg/mL
Chemical Name/SMILES

3-Isoquinolinecarboxamide, 1-(2-fluoro-5-nitrophenyl)-N-methyl-N-(1-methylpropyl)-

References

1. Doble A, et al. Mol Pharmacol. 1987 Jan;31(1):42-9.

2. Doble A, et al. J Recept Res. 1987;7(1-4):55-70.

3. Skowroński R, et al. Eur J Pharmacol. 1988 Mar 29;148(2):187-93.

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