PKC-IN-6c |CAS:2026603-86-9 Probechem Biochemicals

Chemical Structure : PKC-IN-6c

PKC-IN-6c (PKC inhibitor 6c)

Catalog No.: PC-60366Not For Human Use, Lab Use Only.

A novel, potent, brain permeant PKC inhibitor with IC50 of 80 nM, without detectable binding to the estrogen receptor (Ki>10 uM).

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Biological Activity

A novel, potent, brain permeant PKC inhibitor with IC50 of 80 nM, without detectable binding to the estrogen receptor (Ki>10 uM); effectively blocks amphetamine-induced locomotor stimulation, more potently inhibits PKC than tamoxifen and reduces amphetamine-stimulated dopamine efflux.

Physicochemical Properties

M.Wt	565.762
Formula	C35H43N5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3,3-bis(4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)-2-phenylacrylonitrile

References

1. Newman AH, et al. Neuropsychopharmacology. 2017 Jun 8. doi: 10.1038/npp.2017.116.

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PKC-IN-6c (PKC inhibitor 6c)

Biological Activity

Physicochemical Properties

References

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