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PSB-1011

Chemical Structure : PSB-1011

CAS No.: 4499-01-8

PSB-1011 (PSB1011)

Catalog No.: PC-26167Not For Human Use, Lab Use Only.

PSB-1011 is a potent, moderately selective rat P2X2 receptor antagonist with IC50 of 79 nM, weakly inhibits P2X1 and P2X3 receptors and shows no activity against P2X4 and P2X7 receptors.

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    Biological Activity

    PSB-1011 is a potent, moderately selective rat P2X2 receptor antagonist with IC50 of 79 nM, weakly inhibits P2X1 and P2X3 receptors and shows no activity against P2X4 and P2X7 receptors.

    Physicochemical Properties

    M.Wt 681.38
    Formula C23H12Cl2N6Na2O8S2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    sodium 1-amino-4-((3-((4,6-dichloro-1,3,5-triazin-2-yl)amino)-4-sulfonatophenyl)amino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate

    References

    1. Baqi Y, et al. J Med Chem. 2011;54:817–830.

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