PSB-16671 | GPR84 agonist | Probechem Biochemicals

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Chemical Structure : PSB-16671

PSB-16671 (PSB16671)

Catalog No.: PC-72359Not For Human Use, Lab Use Only.

PSB-16671 is a novel orthosteric and allosteric activator of GPR84, activates human GPR84 with EC50 of 41.3 nM in cAMP accumulation assays.

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Biological Activity

PSB-16671 is a novel orthosteric and allosteric activator of GPR84, activates human GPR84 with EC50 of 41.3 nM in cAMP accumulation assays.
PSB-16671 is selective versus related fatty acid receptors and the arylhydrocarbon receptor.
PSB-16671 shows an EC50 of 5.47 uM in β-Arrestin assays, and allosteric KB value of 634 nM.

Physicochemical Properties

M.Wt	318.275
Formula	C17H10F4N2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	di(5,7-difluoro-1H-indole-3-yl)methane

References

1. Sarah J Mancini, et al. Sci Rep. 2019 Feb 12;9(1):1861.
2. Pillaiyar T, et al. J Med Chem. 2017 May 11;60(9):3636-3655.

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PSB-16671 (PSB16671)

Biological Activity

Physicochemical Properties

References

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