PfKRS1 inhibitor 30

Chemical Structure : PfKRS1 inhibitor 30

Catalog No.: PC-27033Not For Human Use, Lab Use Only.

PfKRS1 inhibitor 30 is a potent selective inhibitor of P. falciparum lysyl-tRNA synthetase (PfKRS1) with pIC50 of 6.9, >1,000-fold selectivity for PfKRS1 over the human enzyme, exhibits potency against Pfalciparum (3D7) asexual blood stage with EC50 of 6 nM.

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Biological Activity

Physicochemical Properties

M.Wt	534.55
Formula	C24H32F6N6O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-(((1R,3S)-1-(2-(1,7-diazaspiro[3.5]nonan-7-yl)ethyl)-3-(trifluoromethyl)cyclohexyl)methyl)-2-amino-4-(trifluoromethyl)-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-5-one

References

1. Forte B, et al. J Med Chem. 2026 Jun 2. doi: 10.1021/acs.jmedchem.6c00823.

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