Chemical Structure : Pimelic Diphenylamide 106
CAS No.: 937039-45-7
Catalog No.: PC-45618Not For Human Use, Lab Use Only.
A slow, tight-binding inhibitor of class I HDACs (HDAC1/2/3, Ki=148/102/14 nM respectively).
Packing | Price | Stock | Quantity |
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10 mg | $80 | In stock | |
50 mg | $320 | In stock | |
100 mg | $520 | In stock |
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A slow, tight-binding inhibitor of class I HDACs (HDAC1/2/3, Ki=148/102/14 nM respectively); shows weak inhibition on HDAC8 (IC50=5 uM); has preference toward HDAC3.
M.Wt | 339.4314 | |
Formula | C20H25N3O2 | |
Appearance | Solid | |
Storage |
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Solubility |
DMSO: ≥ 25 mg/mL |
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Chemical Name/SMILES |
Heptanediamide, N1-(2-aminophenyl)-N7-(4-methylphenyl)- |
1. Chou CJ, et al. J Biol Chem. 2008 Dec 19;283(51):35402-9.
2. Xu C, et al. Chem Biol. 2009 Sep 25;16(9):980-9.
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