Chemical Structure : QCA276
Catalog No.: PC-35400Not For Human Use, Lab Use Only.
QCA276 is a novel potent BET proteins inhibitor with IC50/Ki of 10/.3 nM, QCA276 is the BET ligand for PROTAC QCA570.
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QCA276 is a novel potent BET proteins inhibitor with IC50/Ki of 10/.3 nM, QCA276 is the BET ligand for PROTAC QCA570; effectively inhibits human BRD2, BRD3, and BRD4 BD1 and BD2 proteins with Ki of 2-20 nM.
M.Wt | 401.488 | |
Formula | C22H19N5OS | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Qin C, et al. J Med Chem. 2018 Jul 18. doi: 10.1021/acs.jmedchem.8b00506.
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