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Chemical Structure : RLX-33
CAS No.: 2784577-71-3
Catalog No.: PC-38726Not For Human Use, Lab Use Only.
RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $248 | In stock | |
| 10 mg | $398 | In stock | |
| 25 mg | $628 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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RLX-33 is a selective small-molecule nonpeptide antagonist of neuropeptide relaxin-3/RXFP3 with IC50 of 2.36 uM (cAMP functional assays), selective for RXFP3 over RXFP1 and RXFP4.
RLX-33 has favorable pharmacokinetic properties for behavioral assessment.
RLX-33 blocked food intake induced by the RXFP3-selective agonist R3/I5.
| M.Wt | 462.890 | |
| Formula | C24H19ClN4O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-(4-(3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl)phenyl)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxamide |
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1. Elaine A. Gay, et al. J. Med. Chem. 2022, May 20, 2022
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