RTI-348 | CB1 antagonist | Probechem Biochemicals

Chemical Structure : RTI-348

RTI-348 (RTI 348)

Catalog No.: PC-23093Not For Human Use, Lab Use Only.

RTI-348 is a potent, peripherally selective, orally active, and metabolically stable antagonist of cannabinoid receptor 1 (CB1) with Ki of 6.2 nM, 153-fold selective over CB2.

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Biological Activity

RTI-348 is a potent, peripherally selective, orally active, and metabolically stable antagonist of cannabinoid receptor 1 (CB1) with Ki of 6.2 nM, 153-fold selective over CB2.

Physicochemical Properties

M.Wt	593.53
Formula	C29H26Cl2N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(1-(8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl)-4-phenylpiperidin-4-yl)methanesulfonamide

References

1. Lucas T Laudermilk, et al. ACS Pharmacol Transl Sci. 2024 Aug 8;7(9):2856-2868.

2. Alan Fulp, et al. J Med Chem. 2012 Nov 26;55(22):10022-32.

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RTI-348 (RTI 348)

Biological Activity

Physicochemical Properties

References

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