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RTICBM-229

Chemical Structure : RTICBM-229

CAS No.: 2250355-35-0

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RTICBM-229 (RTICBM229)

Catalog No.: PC-72729Not For Human Use, Lab Use Only.

RTICBM-229 is a potent, selective, brain-penetrant CB1 negative allosteric modulator (NAM) with IC50 of 169 nM in Ca2+ assay, 40 nM in GTPγS assay.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

RTICBM-229 is a potent, selective, brain-penetrant CB1 negative allosteric modulator (NAM) with IC50 of 169 nM in Ca2+ assay, 40 nM in GTPγS assay.

Physicochemical Properties

M.Wt 311.769
Formula C17H14ClN3O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-(3-(1H-pyrrol-2-yl)phenyl)-3-(4-chlorophenyl)urea

References

1. Thuy Nguyen, et al. J Med Chem. 2019 Nov 14;62(21):9806-9823.

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