RUVBL1/2 ATPase-IN-1

Chemical Structure : RUVBL1/2 ATPase-IN-1

CAS No.: 423128-55-6

Catalog No.: PC-25732Not For Human Use, Lab Use Only.

RUVBL1/2 ATPase-IN-1 is a small-molecule inhibitor of RUVBL1/2 ATPase with IC50 of 6.0 uM and 7.7 uM against RUVBL1/2 complex and RUVBL1 respectively.

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10 mg	$458	In stock
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Biological Activity

RUVBL1/2 ATPase-IN-1 is a small-molecule inhibitor of RUVBL1/2 ATPase with IC50 of 6.0 uM and 7.7 uM against RUVBL1/2 complex and RUVBL1 respectively.
RUVBL1/2 ATPase-IN-1 shows potent inhibition in cell lines A549, H1795, HCT116, and MDA-MB-231 with IC50 values of 15 ± 1.2 μM, 15 ± 1.8 μM, 11 ± 1.0 μM, and 8.9 ± 0.9 μM respectively.

Physicochemical Properties

M.Wt	507.56
Formula	C28H28F3N5O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(5,7-dimethyl-6-(4-methylbenzyl)pyrazolo[1,5-a]pyrimidin-3-yl)(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)methanone

References

1. Zhang G, et al. Bioorg Med Chem. 2022;62:116726.

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