Chemical Structure : S-2101
CAS No.: 1239262-36-2
Catalog No.: PC-61645Not For Human Use, Lab Use Only.
S-2101 is a potent lysine-specific demethylase 1 (LSD1) inhibitor with Ki of 0.61 uM.
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S-2101 is a potent lysine-specific demethylase 1 (LSD1) inhibitor with Ki of 0.61 uM.
S-2101 displays weaker inhibition to MAO-B and MAO-A compared with Tranylcypromine (2-PCPA).
S-2101 protects against cisplatin-induced hair cell loss by preventing demethylation of histone H3K4 (H3K4me2).
S-2101 induces cytotoxicity in ovarian cancer lines.
M.Wt | 311.75 | |
Formula | C16H15F2NO.HCl | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
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Chemical Name/SMILES |
(1R,2S)-rel-2-[3,5-Difluoro-2-(phenylmethoxy)phenyl]cycloprpanamine hydrochloride |
1. Mimasu S, et al. Biochemistry. 2010 Aug 3;49(30):6494-503.
2. Konovalov S, et al. J Ovarian Res. 2013 Oct 29;6(1):75.
3. He Y, et al. Mol Neurobiol. 2015 Aug;52(1):196-205.
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