Chemical Structure : SB-408124
CAS No.:
288150-92-5
SB-408124
(SB 408124;SB408124)
Catalog No. : PC-45951Not For Human Use, Lab Use Only.
SB-408124 is a potent, selective OX1 receptor (OX1R) antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay).
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4595101
Biological Activity
SB-408124 is a potent, selective OX1 receptor (OX1R ) antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay).
Physicochemical Properties
M.Wt
356.3692
Formula
C19H18F2N4O
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
Urea, N-(6,8-difluoro-2-methyl-4-quinolinyl)-N'-[4-(dimethylamino)phenyl]-
References
1. Langmead CJ, et al. Br J Pharmacol. 2004 Jan;141(2):340-6.
2. Malherbe P, et al. Mol Pharmacol. 2009 Sep;76(3):618-31.
3. Girault EM, et al. Brain Res. 2013 Aug 21;1527:238-45.
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