SGC2085 | CARM1 inhibitor | Probechem Biochemicals

Chemical Structure : SGC2085

CAS No.: 1821908-48-8

SGC2085 (SGC-2085, SGC 2085)

Catalog No.: PC-42198Not For Human Use, Lab Use Only.

SGC2085 is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM, displays >100-fold selectivity over other PRMTs (PRMT6 IC50=5.3 uM).

Packing	Price	Stock
1 mg	$128	In stock
5 mg	$258	In stock
10 mg	$398	In stock
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Biological Activity

SGC2085 is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM, displays >100-fold selectivity over other PRMTs (PRMT6 IC50=5.3 uM).
SGC2085 also shows complete selectivity against a panel of 21 human protein methyltransferases.

Physicochemical Properties

M.Wt	312.4061
Formula	C19H24N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: ≥ 32 mg/mL
Chemical Name/SMILES	Propanamide, 2-amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]-, (2S)-

References

1. Ferreira de Freitas R, et al. J Med Chem. 2016 Jul 28;59(14):6838-47.

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SGC2085 (SGC-2085, SGC 2085)

Biological Activity

Physicochemical Properties

References

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