SGC8158 | PRMT7 inhibitor | Probechem Biochemicals

Chemical Structure : SGC8158

SGC8158 (SGC-8158, SGC 8158)

Catalog No.: PC-72395Not For Human Use, Lab Use Only.

SGC8158 (SGC-8158) is a potent, selective, and SAM-competitive inhibitor of PRMT7 with IC50 of <2.5 nM, the active component of it's cell permeable prodrug SGC3027.

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Biological Activity

SGC8158 (SGC-8158) is a potent, selective, and SAM-competitive inhibitor of PRMT7 with IC50 of <2.5 nM, the active component of it's cell permeable prodrug SGC3027.

Physicochemical Properties

M.Wt	555.094
Formula	C27H31ClN6O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(2R,3R,4S,5S)-2-(6-amino-9H-purin-9-yl)-5-(((4-(((4'-chloro-[1,1'-biphenyl]-3-yl)methyl)amino)butyl)thio)methyl)tetrahydrofuran-3,4-diol

References

1. Szewczyk MM, et al. Nat Commun. 2020 May 14;11(1):2396.

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SGC8158 (SGC-8158, SGC 8158)

Biological Activity

Physicochemical Properties

References

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