SJ830599 |CAS: 2215098-23-8 Probechem Biochemicals

Chemical Structure : SJ830599

SJ830599 (SJ 830599)

Catalog No.: PC-63255Not For Human Use, Lab Use Only.

SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1.

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Biological Activity

SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1; demonstrates cytotoxicity against several pediatric cancer cell lines with EC50 values (HD-MB03 EC50=480 nM) comparable to BET inhibitor (BETi) clinical candidates.

Physicochemical Properties

M.Wt	356.422
Formula	C20H24N2O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Isopropyl ((2S,4R)-1-acetyl-6-(furan-2-yl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)carbamate

References

1. Shadrick WR, et al. Bioorg Med Chem. 2018 Jan 1;26(1):25-36.

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SJ830599 (SJ 830599)

Biological Activity

Physicochemical Properties

References

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