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SMYD3 inhibitor 49

Chemical Structure : SMYD3 inhibitor 49

CAS No.: 2411394-32-4

SMYD3 inhibitor 49

Catalog No.: PC-49814Not For Human Use, Lab Use Only.

SMYD3 inhibitor 49 is a potent and selective SMYD3 inhibitor with IC50 of 6.3 and 44 nM in biochemical and cellular MEKK2me assays, respectively.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

SMYD3 inhibitor 49 is a potent and selective SMYD3 inhibitor with IC50 of 6.3 and 44 nM in biochemical and cellular MEKK2me assays, respectively.

Physicochemical Properties

M.Wt 506.59
Formula C22H33F3N4O4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

5-cyclopropyl-N-(1-(((1r,4r)-4-((4,4,4-trifluorobutyl)amino)cyclohexyl)sulfonyl)piperidin-4-yl)isoxazole-3-carboxamide

References

1. Dai-Shi Su, et al. ACS Med Chem Lett. 2019 Dec 27;11(2):133-140.

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