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SNT-207858

Chemical Structure : SNT-207858

CAS No.: 1104662-66-9

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SNT-207858 (SNT207858)

Catalog No.: PC-49761Not For Human Use, Lab Use Only.

SNT-207858 (SNT207858) is a potent, selective, BBB-penetrating, and orally active melanocortin-4 (MC4R) receptor antagonist with binding/fuaction IC50 of 22/11 nM, respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    SNT-207858 (SNT207858) is a potent, selective, BBB-penetrating, and orally active melanocortin-4 (MC4R) receptor antagonist with binding/fuaction IC50 of 22/11 nM, respectively.
    SNT-207858 treatment increase food intake in healthy mice.
    SNT-207858 prevented tumor induced weight loss, and diminished loss of lean body mass and fat mass.

    Physicochemical Properties

    M.Wt 616.63
    Formula C32H43Cl2N5O3
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-((R)-3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((R)-2-(pyrrolidin-1-yl)butoxy)pyridin-2-yl)piperidin-1-yl)propan-2-yl)pyrrolidine-1-carboxamide

    References

    1. Weyermann P, et al. PLoS One. 2009;4(3):e4774.

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